Iptakalim Hydrochloride
CAS No. 642407-63-4
Iptakalim Hydrochloride ( —— )
Catalog No. M27888 CAS No. 642407-63-4
Iptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well as an α4β2-containing nicotinic acetylcholine receptor (nAChR) antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 43 | Get Quote |
|
10MG | 67 | Get Quote |
|
25MG | 133 | Get Quote |
|
50MG | 217 | Get Quote |
|
100MG | 327 | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
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Product NameIptakalim Hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionIptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well as an α4β2-containing nicotinic acetylcholine receptor (nAChR) antagonist.
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DescriptionIptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well as an α4β2-containing nicotinic acetylcholine receptor (nAChR) antagonist. Iptakalim is also a K(ir) 6.1/SUR2B activator that can attenuate hypoxia-induced pulmonary arterial hypertension in rats by endothelial function protection.
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetPotassium Channel
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RecptorAldose reductase
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Research Area——
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Indication——
Chemical Information
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CAS Number642407-63-4
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Formula Weight179.7
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Molecular FormulaC9H22ClN
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Purity>98% (HPLC)
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Solubility——
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SMILESCl.CC(C)NC(C)(C)C(C)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Simard-Duquesne N, et al. The effects of a new aldose reductase inhibitor (tolrestat) in galactosemic and diabetic rats. Metabolism. 1985 Oct;34(10):885-92.
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